Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
SL0101-1 C25H24O12 516.46 RSK Smith (2005) Cancer Res. 65 1027 Goden Sayeski (2006) Am. J. Cell. Physiol. 291 1308 Tocris Download

Results as Barchart

View results as a bar chart
10µM

Results as Table

Screening Concentration: 10µM
Kinase % Activity Remaining Standard Deviation
MKK1 88 7
ERK1 98 5
ERK2 98 9
JNK1 94 9
JNK2 94 7
JNK3 97 2
p38 alpha MAPK 94 8
p38 beta MAPK 98 1
p38 gamma MAPK 103 8
p38 delta MAPK 88 10
ERK8 89 9
RSK1 23 1
RSK2 30 5
PDK1 102 8
PKB alpha 88 7
PKB beta 98 4
SGK1 109 10
S6K1 103 8
PKA 92 7
ROCK 2 109 4
PRK2 106 7
PKC alpha 90 6
PKC zeta 81 2
PKD1 88 3
MSK1 101 1
MNK1 82 0
MNK2 96 6
MAPKAP-K2 95 3
MAPKAP-K3 111 12
PRAK 82 3
CAMKK alpha 116 9
CAMKK beta 107 7
CAMK1 105 7
SmMLCK 109 4
PHK 96 5
CHK1 82 0
CHK2 98 2
GSK3 beta 87 11
CDK2-Cyclin A 106 5
PLK1 111 11
Aurora B 45 6
Aurora C 76 2
AMPK 88 0
MARK3 112 6
BRSK2 80 4
MELK 102 6
CK1 delta 87 1
CK2 101 6
DYRK1A 79 6
DYRK2 89 4
DYRK3 84 3
NEK2a 101 8
NEK6 108 13
NEK7 104 0
IKK beta 99 2
PIM1 71 2
PIM2 95 1
PIM3 49 2
SRPK1 95 4
EF2K 85 4
HIPK2 72 8
HIPK3 109 7
PAK4 95 5
PAK5 85 5
PAK6 126 9
MST2 98 1
Src 104 3
Lck 88 0
CSK 105 6

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