Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
Rapamycin C51H79NO13 914.2 p70S6K Powell D.J. (2003) Mol. Cell Biol. 23 7794 Braun W. (1995) FASEB J. 9 63 Merck (Calbiochem) Download

Results as Barchart

View results as a bar chart
1µM

Results as Table

Screening Concentration: 1µM
Kinase % Activity Remaining Standard Deviation
MKK1 93 4
ERK1 100 1
ERK2 93 4
JNK1 90 8
JNK2 81 0
JNK3 80 0
p38 alpha MAPK 74 4
p38 beta MAPK 83 0
p38 gamma MAPK 80 7
p38 delta MAPK 92 4
ERK8 96 5
RSK1 90 3
RSK2 97 5
PDK1 84 0
PKB alpha 91 3
PKB beta 84 9
SGK1 93 1
S6K1 105 7
PKA 77 1
ROCK 2 103 3
PRK2 78 1
PKC alpha 88 3
PKC zeta 92 5
PKD1 92 2
MSK1 85 2
MNK1 83 1
MNK2 101 3
MAPKAP-K2 108 4
MAPKAP-K3 104 4
PRAK 91 2
CAMKK alpha 80 8
CAMKK beta 82 1
CAMK1 97 0
SmMLCK 107 1
PHK 95 2
CHK1 97 6
CHK2 92 2
GSK3 beta 83 5
CDK2-Cyclin A 92 3
PLK1 78 3
Aurora B 86 5
Aurora C 97 5
AMPK 87 2
MARK3 88 3
BRSK2 90 4
MELK 74 4
CK1 delta 88 1
CK2 92 9
DYRK1A 91 1
DYRK2 83 8
DYRK3 87 1
NEK2a 82 5
NEK6 95 3
NEK7 102 5
IKK beta 82 3
PIM1 91 2
PIM2 117 0
PIM3 88 1
SRPK1 84 1
EF2K 94 0
HIPK2 93 6
HIPK3 108 4
PAK4 81 1
PAK5 89 8
PAK6 88 1
MST2 90 5
Src 85 0
Lck 79 6
CSK 83 1

Do you need any help? Please get in touch and we’ll be happy to lend a hand.