Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
LiCl ClLi 42.394 GSK3b Galli C. (2013) Clin Oral Implants Res. 921-7. WO2001074164 Sigma Download

Results as Barchart

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Results as Table

Screening Concentration:
Kinase % Activity Remaining Standard Deviation
MKK1 18 7
MKK1 83 8
ERK1 92 3
ERK1 101 6
ERK2 60 5
ERK2 71 7
JNK1 76 10
JNK1 81 4
JNK2 107 14
JNK2 85 8
JNK3 77 0
JNK3 77 4
p38 alpha MAPK 111 12
p38 alpha MAPK 100 8
p38 beta MAPK 113 10
p38 beta MAPK 102 2
p38 gamma MAPK 70 4
p38 gamma MAPK 90 1
p38 delta MAPK 78 13
p38 delta MAPK 47 4
ERK8 75 5
ERK8 61 5
RSK1 80 8
RSK1 54 0
RSK2 57 8
RSK2 58 2
PDK1 75 4
PDK1 84 7
PKB alpha 72 14
PKB alpha 77 5
PKB beta 84 7
PKB beta 77 6
SGK1 109 10
SGK1 119 7
S6K1 132 6
S6K1 127 14
PKA 64 3
PKA 76 5
ROCK 2 115 7
ROCK 2 109 14
PRK2 77 8
PRK2 86 8
PKC alpha 73 3
PKC alpha 90 9
PKC zeta 59 4
PKC zeta 72 2
PKD1 92 5
PKD1 95 3
MSK1 79 8
MSK1 85 6
MNK1 53 8
MNK1 46 6
MNK2 56 3
MNK2 35 8
MAPKAP-K2 76 7
MAPKAP-K2 56 3
MAPKAP-K3 92 12
MAPKAP-K3 71 2
PRAK 56 13
PRAK 75 4
CAMKK beta 104 8
CAMK1 62 0
CAMK1 79 4
SmMLCK 35 2
SmMLCK 43 6
PHK 26 8
PHK 60 2
CHK1 61 5
CHK1 72 5
CHK2 43 3
CHK2 59 8
GSK3 beta 25 7
GSK3 beta 30 4
CDK2-Cyclin A 79 5
CDK2-Cyclin A 100 1
PLK1 24 3
PLK1 75 4
Aurora B 24 2
Aurora B 57 2
Aurora C 45 0
Aurora C 60 2
AMPK 103 7
AMPK 101 15
MARK3 89 6
MARK3 71 2
BRSK2 81 7
BRSK2 60 5
MELK 82 5
MELK 81 8
CK1 delta 55 10
CK1 delta 44 6
CK2 49 4
CK2 86 4
DYRK1A 89 5
DYRK1A 89 4
DYRK2 106 4
DYRK2 94 6
DYRK3 102 14
DYRK3 88 8
NEK2a 78 6
NEK2a 74 8
NEK6 70 3
NEK6 53 12
NEK7 58 1
NEK7 73 6
IKK beta 70 1
IKK beta 88 10
IKK epsilon 51 8
IKK epsilon 31 12
TBK1 54 5
TBK1 59 8
PIM1 76 2
PIM1 68 1
PIM2 120 3
PIM2 120 6
PIM3 58 3
PIM3 97 2
SRPK1 85 12
SRPK1 95 5
EF2K 58 6
EF2K 38 10
HIPK2 66 6
HIPK2 38 2
HIPK3 50 8
HIPK3 22 0
PAK4 91 5
PAK4 81 6
PAK5 74 3
PAK5 81 9
PAK6 73 8
PAK6 89 2
MST2 94 5
MST2 98 6
MST4 69 2
MST4 81 3
Src 78 7
Src 62 4
Lck 52 9
Lck 76 10
CSK 70 5
CSK 89 2
YES1 64 5
YES1 33 6
SYK 92 3
SYK 70 1
EPH-A2 71 1
EPH-A2 77 4
FGF-R1 35 2
FGF-R1 53 3
IRR 82 5
IRR 94 7

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