Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
KT5720 C32H31N3O5 537.6 PKA Simpson CS. Morris BJ. (1995) Neuroscience 68 97-106 Cabell L. Audesirk G. (1993) Int. J. Dev. Neurosci. 11 357 US20100216703 Merck (Calbiochem) Download

Results as Barchart

View results as a bar chart
1µM

Results as Table

Screening Concentration: 1µM
Kinase % Activity Remaining Standard Deviation
MKK1 24 2
ERK1 79 0
ERK2 66 1
JNK1 38 0
JNK2 63 1
JNK3 43 0
p38 alpha MAPK 96 4
p38 beta MAPK 90 2
p38 gamma MAPK 69 5
p38 delta MAPK 111 4
ERK8 57 2
RSK1 18 0
RSK2 19 6
PDK1 3 0
PKB alpha 91 4
PKB beta 82 6
SGK1 20 0
S6K1 93 9
PKA 50 8
ROCK 2 85 1
PRK2 10 2
PKC alpha 60 8
PKC zeta 106 3
PKD1 12 4
MSK1 39 1
MNK1 61 0
MNK2 13 3
MAPKAP-K2 28 1
MAPKAP-K3 98 1
PRAK 71 6
CAMKK alpha 60 1
CAMKK beta 27 0
CAMK1 76 6
SmMLCK 54 5
PHK 5 0
CHK1 18 1
CHK2 59 6
GSK3 beta 76 4
CDK2-Cyclin A 65 1
PLK1 81 0
Aurora B 14 4
Aurora C 15 0
AMPK 15 2
MARK3 29 2
BRSK2 14 2
MELK 14 1
CK1 delta 97 2
CK2 84 1
DYRK1A 38 8
DYRK2 66 1
DYRK3 40 7
NEK2a 79 4
NEK6 99 6
NEK7 102 8
IKK beta 62 7
PIM1 40 0
PIM2 67 5
PIM3 7 0
SRPK1 69 4
EF2K 95 0
HIPK2 77 3
HIPK3 112 0
PAK4 36 4
PAK5 62 7
PAK6 70 2
MST2 26 4
Src 78 5
Lck 59 7
CSK 67 1

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