Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
KN62 C38H35N5O6S2 721.9 CaMKII Minami H. (1994) Biochem. Biophys. Res. Commun. 199 241 US20080255244 Merck (Calbiochem) Download

Results as Barchart

View results as a bar chart
10µM

Results as Table

Screening Concentration: 10µM
Kinase % Activity Remaining Standard Deviation
MKK1 93 8
ERK1 102 6
ERK2 92 3
JNK1 110 2
JNK2 89 2
JNK3 79 0
p38 alpha MAPK 91 3
p38 beta MAPK 84 2
p38 gamma MAPK 102 1
p38 delta MAPK 90 9
ERK8 99 1
RSK1 116 3
RSK2 60 2
PDK1 99 0
PKB alpha 75 0
PKB beta 83 5
SGK1 75 1
S6K1 61 1
PKA 76 2
ROCK 2 87 1
PRK2 87 4
PKC alpha 93 5
PKC zeta 99 2
PKD1 87 0
MSK1 81 1
MNK1 103 5
MNK2 101 1
MAPKAP-K2 56 4
MAPKAP-K3 74 5
PRAK 45 1
CAMKK alpha 85 6
CAMKK beta 88 0
CAMK1 38 4
SmMLCK 80 1
PHK 87 1
CHK1 120 11
CHK2 123 1
GSK3 beta 58 3
CDK2-Cyclin A 105 8
PLK1 95 2
Aurora B 89 1
Aurora C 91 1
AMPK 115 1
MARK3 90 6
BRSK2 96 5
MELK 76 7
CK1 delta 93 8
CK2 105 3
DYRK1A 38 7
DYRK2 76 0
DYRK3 81 1
NEK2a 90 8
NEK6 74 2
NEK7 91 3
IKK beta 63 2
PIM1 53 0
PIM2 87 1
PIM3 61 2
SRPK1 70 2
EF2K 130 1
HIPK2 99 3
HIPK3 107 6
PAK4 89 8
PAK5 104 3
PAK6 113 2
MST2 102 3
Src 94 4
Lck 30 0
CSK 79 0

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