Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
Kenpaullone C16H11BrN2O 327.2 GSK, CDK Bain J. (2003) Biochem. J. 371 199 Buolamwini J.K. (2000) Curr. Pharm. Des. 6 379 WO2013184591 Merck (Calbiochem) Download

Results as Barchart

View results as a bar chart
1µM

Results as Table

Screening Concentration: 1µM
Kinase % Activity Remaining Standard Deviation
MKK1 88 2
ERK1 85 7
ERK2 88 8
JNK1 89 2
JNK2 83 2
JNK3 84 0
p38 alpha MAPK 94 5
p38 beta MAPK 95 0
p38 gamma MAPK 86 5
p38 delta MAPK 92 7
ERK8 75 6
RSK1 83 3
RSK2 83 8
PDK1 62 3
PKB alpha 94 6
PKB beta 90 6
SGK1 80 0
S6K1 113 2
PKA 63 4
ROCK 2 42 5
PRK2 57 5
PKC alpha 87 6
PKC zeta 71 6
PKD1 86 1
MSK1 88 1
MNK1 85 2
MNK2 102 1
MAPKAP-K2 91 6
MAPKAP-K3 97 1
PRAK 79 1
CAMKK alpha 74 5
CAMKK beta 61 2
CAMK1 87 5
SmMLCK 83 1
PHK 18 1
CHK1 72 5
CHK2 28 2
GSK3 beta 3 0
CDK2-Cyclin A 14 0
PLK1 90 1
Aurora B 49 4
Aurora C 83 1
AMPK 94 0
MARK3 36 5
BRSK2 41 0
MELK 55 6
CK1 delta 98 1
CK2 78 5
DYRK1A 80 4
DYRK2 73 5
DYRK3 81 4
NEK2a 87 1
NEK6 93 1
NEK7 97 7
IKK beta 76 4
PIM1 48 0
PIM2 80 1
PIM3 28 0
SRPK1 92 4
EF2K 110 1
HIPK2 81 9
HIPK3 95 0
PAK4 7 0
PAK5 13 2
PAK6 39 5
MST2 41 2
Src 38 1
Lck 29 3
CSK 77 5

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