Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
Harmane C12H10N2 182.22 serotonin, monoamine oxidase Smith KL. (2013) J Psychopharmacol. 162-70 US5256533 Sigma Download

Results as Barchart

View results as a bar chart
1µM

Results as Table

Screening Concentration: 1µM
Kinase % Activity Remainingsort descending Standard Deviation
DYRK1A 44 3
ERK8 69 0
DYRK3 72 3
p38 alpha MAPK 74 1
IKK beta 76 8
NEK2a 78 0
PIM3 80 0
SRPK1 80 2
MST2 80 1
PLK1 80 2
CSK 81 5
MNK1 82 1
MELK 82 2
DYRK2 83 5
Src 83 2
PRAK 84 8
CK2 84 7
JNK2 84 5
PRK2 84 5
CAMKK alpha 85 5
PIM2 85 1
Aurora C 86 2
SGK1 86 4
PKD1 87 1
p38 delta MAPK 89 1
PDK1 89 7
JNK3 89 2
PKC zeta 89 2
MKK1 90 5
CAMK1 90 3
NEK6 90 1
PKC alpha 90 5
p38 beta MAPK 90 7
MSK1 90 11
PKB beta 91 7
CHK2 91 3
CAMKK beta 92 4
JNK1 92 3
Lck 93 1
PIM1 93 1
RSK2 94 1
S6K1 94 3
PKA 94 2
ERK2 95 6
p38 gamma MAPK 96 9
PAK5 97 8
RSK1 98 0
CK1 delta 98 6
CHK1 98 3
BRSK2 100 1
EF2K 100 3
SmMLCK 100 3
PHK 102 3
CDK2-Cyclin A 102 6
MAPKAP-K3 103 6
PKB alpha 103 2
PAK4 103 5
HIPK2 104 5
HIPK3 104 0
PAK6 104 3
ROCK 2 104 1
NEK7 104 0
Aurora B 105 2
ERK1 106 0
GSK3 beta 108 1
MAPKAP-K2 109 3
MNK2 111 4
AMPK 111 12
MARK3 128 3

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