Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
Harmane C12H10N2 182.22 serotonin, monoamine oxidase Smith KL. (2013) J Psychopharmacol. 162-70 US5256533 Sigma Download

Results as Barchart

View results as a bar chart
1µM

Results as Table

Screening Concentration: 1µM
Kinase % Activity Remaining Standard Deviation
MKK1 90 5
ERK1 106 0
ERK2 95 6
JNK1 92 3
JNK2 84 5
JNK3 89 2
p38 alpha MAPK 74 1
p38 beta MAPK 90 7
p38 gamma MAPK 96 9
p38 delta MAPK 89 1
ERK8 69 0
RSK1 98 0
RSK2 94 1
PDK1 89 7
PKB alpha 103 2
PKB beta 91 7
SGK1 86 4
S6K1 94 3
PKA 94 2
ROCK 2 104 1
PRK2 84 5
PKC alpha 90 5
PKC zeta 89 2
PKD1 87 1
MSK1 90 11
MNK1 82 1
MNK2 111 4
MAPKAP-K2 109 3
MAPKAP-K3 103 6
PRAK 84 8
CAMKK alpha 85 5
CAMKK beta 92 4
CAMK1 90 3
SmMLCK 100 3
PHK 102 3
CHK1 98 3
CHK2 91 3
GSK3 beta 108 1
CDK2-Cyclin A 102 6
PLK1 80 2
Aurora B 105 2
Aurora C 86 2
AMPK 111 12
MARK3 128 3
BRSK2 100 1
MELK 82 2
CK1 delta 98 6
CK2 84 7
DYRK1A 44 3
DYRK2 83 5
DYRK3 72 3
NEK2a 78 0
NEK6 90 1
NEK7 104 0
IKK beta 76 8
PIM1 93 1
PIM2 85 1
PIM3 80 0
SRPK1 80 2
EF2K 100 3
HIPK2 104 5
HIPK3 104 0
PAK4 103 5
PAK5 97 8
PAK6 104 3
MST2 80 1
Src 83 2
Lck 93 1
CSK 81 5

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