Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
Harmalol C12H12N2O • HCl • 2H2O 272.73 serotonin, monoamine oxidase Riba J. (2012) Drug Test. 610-6. US5256533 Sigma Download

Results as Barchart

View results as a bar chart
1µM

Results as Table

Screening Concentration: 1µM
Kinase % Activity Remainingsort descending Standard Deviation
ERK8 62 3
DYRK1A 67 6
DYRK3 71 2
PIM3 71 0
IKK beta 73 1
MELK 76 0
PKB beta 81 1
NEK2a 82 4
PLK1 82 0
CSK 83 6
RSK2 83 7
PRAK 84 2
CHK1 84 5
SGK1 85 2
Src 85 5
MKK1 86 1
DYRK2 86 4
PRK2 86 2
PHK 87 3
PKC zeta 87 0
PKB alpha 88 1
GSK3 beta 88 3
SRPK1 88 8
MAPKAP-K2 88 1
p38 delta MAPK 89 4
CAMKK beta 90 1
CK2 90 0
PKA 90 3
ROCK 2 90 7
Aurora B 90 7
Aurora C 90 5
MST2 90 3
PAK6 91 1
PKC alpha 91 1
PIM1 91 1
PDK1 92 5
Lck 92 1
CK1 delta 93 9
HIPK3 93 8
NEK6 93 1
S6K1 94 8
ERK2 94 5
PAK5 95 4
p38 beta MAPK 95 3
MSK1 95 1
p38 alpha MAPK 96 2
MNK1 97 1
MAPKAP-K3 98 9
BRSK2 98 4
JNK2 99 6
RSK1 99 9
HIPK2 100 1
CDK2-Cyclin A 100 1
PIM2 100 1
CAMK1 101 3
EF2K 101 6
CAMKK alpha 102 1
JNK1 102 3
PAK4 104 6
p38 gamma MAPK 104 1
ERK1 106 0
MNK2 106 5
SmMLCK 107 9
NEK7 108 7
AMPK 109 1
PKD1 110 2
JNK3 112 0
CHK2 121 1
MARK3 131 8

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