Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
Harmalol C12H12N2O • HCl • 2H2O 272.73 serotonin, monoamine oxidase Riba J. (2012) Drug Test. 610-6. US5256533 Sigma Download

Results as Barchart

View results as a bar chart
1µM

Results as Table

Screening Concentration: 1µM
Kinase % Activity Remaining Standard Deviation
MKK1 86 1
ERK1 106 0
ERK2 94 5
JNK1 102 3
JNK2 99 6
JNK3 112 0
p38 alpha MAPK 96 2
p38 beta MAPK 95 3
p38 gamma MAPK 104 1
p38 delta MAPK 89 4
ERK8 62 3
RSK1 99 9
RSK2 83 7
PDK1 92 5
PKB alpha 88 1
PKB beta 81 1
SGK1 85 2
S6K1 94 8
PKA 90 3
ROCK 2 90 7
PRK2 86 2
PKC alpha 91 1
PKC zeta 87 0
PKD1 110 2
MSK1 95 1
MNK1 97 1
MNK2 106 5
MAPKAP-K2 88 1
MAPKAP-K3 98 9
PRAK 84 2
CAMKK alpha 102 1
CAMKK beta 90 1
CAMK1 101 3
SmMLCK 107 9
PHK 87 3
CHK1 84 5
CHK2 121 1
GSK3 beta 88 3
CDK2-Cyclin A 100 1
PLK1 82 0
Aurora B 90 7
Aurora C 90 5
AMPK 109 1
MARK3 131 8
BRSK2 98 4
MELK 76 0
CK1 delta 93 9
CK2 90 0
DYRK1A 67 6
DYRK2 86 4
DYRK3 71 2
NEK2a 82 4
NEK6 93 1
NEK7 108 7
IKK beta 73 1
PIM1 91 1
PIM2 100 1
PIM3 71 0
SRPK1 88 8
EF2K 101 6
HIPK2 100 1
HIPK3 93 8
PAK4 104 6
PAK5 95 4
PAK6 91 1
MST2 90 3
Src 85 5
Lck 92 1
CSK 83 6

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