Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
Harmaline C13H14N2O 214.263 serotonin, monoamine oxidase Herraiz T. (2013) Drug Test. 1002/dta.1530. WO1999041984 Sigma Download

Results as Barchart

View results as a bar chart
1µM

Results as Table

Screening Concentration: 1µM
Kinase % Activity Remainingsort descending Standard Deviation
DYRK1A 29 4
ERK8 44 4
DYRK3 49 5
CK1 delta 65 5
PRAK 73 1
DYRK2 73 1
ROCK 2 78 6
PLK1 79 1
MNK1 80 0
Lck 81 1
CSK 81 6
PAK5 83 6
PHK 83 6
PKC zeta 83 2
PDK1 85 8
SGK1 85 7
JNK2 85 6
PRK2 85 1
ERK2 86 0
CK2 87 1
p38 alpha MAPK 87 4
CAMKK beta 88 7
PKA 88 1
JNK3 88 0
SRPK1 89 5
MAPKAP-K2 89 4
Aurora B 89 4
PIM3 90 6
HIPK2 90 1
PAK4 90 1
PKC alpha 90 8
p38 delta MAPK 92 5
MNK2 92 2
CAMKK alpha 92 1
p38 beta MAPK 92 0
S6K1 93 1
CHK1 93 4
MSK1 93 1
PKB alpha 94 0
MKK1 94 2
Src 94 5
NEK6 94 1
IKK beta 94 4
MELK 95 0
JNK1 95 3
NEK2a 96 6
MAPKAP-K3 97 4
HIPK3 97 0
Aurora C 99 8
GSK3 beta 100 9
CDK2-Cyclin A 100 6
MST2 101 0
BRSK2 103 1
CAMK1 103 0
PIM1 104 6
AMPK 105 1
PKB beta 105 1
PAK6 105 2
EF2K 107 2
ERK1 107 4
NEK7 107 8
PKD1 107 1
RSK1 109 5
MARK3 110 5
SmMLCK 111 2
RSK2 112 0
CHK2 116 5
PIM2 117 1
p38 gamma MAPK 119 5

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