Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
Harmaline C13H14N2O 214.263 serotonin, monoamine oxidase Herraiz T. (2013) Drug Test. 1002/dta.1530. WO1999041984 Sigma Download

Results as Barchart

View results as a bar chart
1µM

Results as Table

Screening Concentration: 1µM
Kinase % Activity Remaining Standard Deviation
MKK1 94 2
ERK1 107 4
ERK2 86 0
JNK1 95 3
JNK2 85 6
JNK3 88 0
p38 alpha MAPK 87 4
p38 beta MAPK 92 0
p38 gamma MAPK 119 5
p38 delta MAPK 92 5
ERK8 44 4
RSK1 109 5
RSK2 112 0
PDK1 85 8
PKB alpha 94 0
PKB beta 105 1
SGK1 85 7
S6K1 93 1
PKA 88 1
ROCK 2 78 6
PRK2 85 1
PKC alpha 90 8
PKC zeta 83 2
PKD1 107 1
MSK1 93 1
MNK1 80 0
MNK2 92 2
MAPKAP-K2 89 4
MAPKAP-K3 97 4
PRAK 73 1
CAMKK alpha 92 1
CAMKK beta 88 7
CAMK1 103 0
SmMLCK 111 2
PHK 83 6
CHK1 93 4
CHK2 116 5
GSK3 beta 100 9
CDK2-Cyclin A 100 6
PLK1 79 1
Aurora B 89 4
Aurora C 99 8
AMPK 105 1
MARK3 110 5
BRSK2 103 1
MELK 95 0
CK1 delta 65 5
CK2 87 1
DYRK1A 29 4
DYRK2 73 1
DYRK3 49 5
NEK2a 96 6
NEK6 94 1
NEK7 107 8
IKK beta 94 4
PIM1 104 6
PIM2 117 1
PIM3 90 6
SRPK1 89 5
EF2K 107 2
HIPK2 90 1
HIPK3 97 0
PAK4 90 1
PAK5 83 6
PAK6 105 2
MST2 101 0
Src 94 5
Lck 81 1
CSK 81 6

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