Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
Gö 6976 C24H18N4O 378.4 PKC Gschwendt M. (1996) FEBS Lett. 392 77 Wenzel-Seifert K. (1994) Biochem. Biophys. Res. Commun. 200 1536 WO2003009809 Merck (Calbiochem) Download

Results as Barchart

View results as a bar chart
0.1µM

Results as Table

Screening Concentration: 0.1µM
Kinase % Activity Remainingsort descending Standard Deviation
MST2 0 0
PHK 1 1
CHK1 1 0
PKC alpha 1 0
PRK2 4 2
PIM3 5 0
RSK2 5 0
PAK4 5 0
PKD1 6 0
PAK5 7 0
MSK1 7 0
PAK6 8 0
RSK1 9 2
CDK2-Cyclin A 10 0
PDK1 11 0
S6K1 16 0
AMPK 16 3
MARK3 16 1
CAMKK beta 16 4
MELK 17 2
PIM1 21 1
Aurora B 23 0
GSK3 beta 24 4
Aurora C 26 3
HIPK2 27 3
SmMLCK 31 1
DYRK1A 33 6
DYRK3 33 6
MNK2 34 0
ERK8 36 4
CAMKK alpha 37 4
ERK2 46 2
BRSK2 48 6
MKK1 50 1
Lck 53 6
CHK2 53 3
JNK1 58 2
HIPK3 58 2
SGK1 59 5
ROCK 2 59 4
ERK1 60 7
DYRK2 60 8
PKA 64 5
PIM2 65 3
MNK1 69 0
JNK3 70 0
Src 74 2
CSK 74 3
IKK beta 76 0
p38 delta MAPK 78 1
JNK2 79 0
PKC zeta 80 4
PLK1 80 1
p38 gamma MAPK 83 8
PRAK 83 3
NEK2a 84 1
PKB alpha 85 1
PKB beta 87 1
CK1 delta 88 3
CK2 88 4
SRPK1 92 5
NEK6 97 6
CAMK1 99 3
MAPKAP-K3 104 7
NEK7 108 1
EF2K 109 3
p38 alpha MAPK 116 4
MAPKAP-K2 118 3
p38 beta MAPK 125 5

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