Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
Gö 6976 C24H18N4O 378.4 PKC Gschwendt M. (1996) FEBS Lett. 392 77 Wenzel-Seifert K. (1994) Biochem. Biophys. Res. Commun. 200 1536 WO2003009809 Merck (Calbiochem) Download

Results as Barchart

View results as a bar chart
0.1µM

Results as Table

Screening Concentration: 0.1µM
Kinase % Activity Remaining Standard Deviation
MKK1 50 1
ERK1 60 7
ERK2 46 2
JNK1 58 2
JNK2 79 0
JNK3 70 0
p38 alpha MAPK 116 4
p38 beta MAPK 125 5
p38 gamma MAPK 83 8
p38 delta MAPK 78 1
ERK8 36 4
RSK1 9 2
RSK2 5 0
PDK1 11 0
PKB alpha 85 1
PKB beta 87 1
SGK1 59 5
S6K1 16 0
PKA 64 5
ROCK 2 59 4
PRK2 4 2
PKC alpha 1 0
PKC zeta 80 4
PKD1 6 0
MSK1 7 0
MNK1 69 0
MNK2 34 0
MAPKAP-K2 118 3
MAPKAP-K3 104 7
PRAK 83 3
CAMKK alpha 37 4
CAMKK beta 16 4
CAMK1 99 3
SmMLCK 31 1
PHK 1 1
CHK1 1 0
CHK2 53 3
GSK3 beta 24 4
CDK2-Cyclin A 10 0
PLK1 80 1
Aurora B 23 0
Aurora C 26 3
AMPK 16 3
MARK3 16 1
BRSK2 48 6
MELK 17 2
CK1 delta 88 3
CK2 88 4
DYRK1A 33 6
DYRK2 60 8
DYRK3 33 6
NEK2a 84 1
NEK6 97 6
NEK7 108 1
IKK beta 76 0
PIM1 21 1
PIM2 65 3
PIM3 5 0
SRPK1 92 5
EF2K 109 3
HIPK2 27 3
HIPK3 58 2
PAK4 5 0
PAK5 7 0
PAK6 8 0
MST2 0 0
Src 74 2
Lck 53 6
CSK 74 3

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