Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
GF 109203X (Go 6850) C25H24N4O2 412.5 PKC Hers I. (1999) FEBS Lett. 460 433 Ku W.-C. (1997) Biochem. Biophys. Res. Commun. 241 730 US7067144 Merck (Calbiochem) Download

Results as Barchart

View results as a bar chart
10µM

Results as Table

Screening Concentration: 10µM
Kinase % Activity Remaining Standard Deviation
MKK1 47 9
ERK2 75 1
JNK1 58 4
p38 alpha MAPK 73 8
p38 beta MAPK 81 3
p38 gamma MAPK 90 2
p38 delta MAPK 102 5
RSK1 0 1
PKB alpha 23 0
SGK1 1 4
S6K1 3 0
PKA 23 6
ROCK 2 43 10
PKC alpha 0 1
PKD1 5 1
MSK1 0 3
MAPKAP-K2 20 1
PRAK 69 3
PHK 0 2
CHK1 6 1
GSK3 beta 2 0
CDK2-Cyclin A 2 4
AMPK 4 4
CK1 delta 83 7
CK2 78 5
DYRK1A 0 3
NEK6 108 4
Lck 27 7
CSK 79 17

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