Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
FMK (Caspase Inhibitor I) C22H30FN3O7 467.5 Caspase Martin U. (2007) Apoptosis 12 525 Misaghi S. (2004) Chem. Biol. 11 1677 WO2001058526 Merck (Calbiochem) Download

Results as Barchart

View results as a bar chart
3µM

Results as Table

Screening Concentration: 3µM
Kinase % Activity Remainingsort descending Standard Deviation
Lck 10 1
Src 10 1
S6K1 33 2
MNK1 42 2
CAMKK beta 49 3
BRSK2 53 6
CSK 55 7
PIM3 56 6
ERK8 58 4
Aurora B 59 3
PIM1 61 6
CK1 delta 63 6
GSK3 beta 65 6
MNK2 65 6
MELK 65 8
DYRK3 68 7
CAMKK alpha 70 12
p38 alpha MAPK 72 2
RSK2 74 2
MSK1 75 3
Aurora C 75 6
MST2 76 4
CAMK1 77 9
AMPK 79 4
HIPK2 79 11
HIPK3 79 9
ERK2 79 5
CDK2-Cyclin A 80 7
MARK3 80 3
MKK1 80 8
JNK1 81 3
CHK2 81 9
PLK1 82 5
PKB alpha 82 3
SmMLCK 82 4
JNK2 83 5
PRK2 83 3
PKD1 83 4
PKC alpha 85 7
p38 beta MAPK 85 4
PIM2 85 10
SRPK1 85 1
PKA 85 7
ROCK 2 86 7
DYRK1A 86 11
CHK1 88 4
PAK5 88 6
JNK3 89 4
PDK1 89 10
NEK6 90 4
PKC zeta 91 5
PAK4 91 1
DYRK2 91 8
NEK7 92 8
IKK beta 92 8
p38 gamma MAPK 92 7
RSK1 92 6
MAPKAP-K3 92 6
CK2 92 10
ERK1 92 6
PAK6 93 5
PHK 93 5
MAPKAP-K2 94 10
NEK2a 95 4
EF2K 97 8
PRAK 97 5
PKB beta 97 4
p38 delta MAPK 103 9
SGK1 107 8

Do you need any help? Please get in touch and we’ll be happy to lend a hand.