Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
FMK (Caspase Inhibitor I) C22H30FN3O7 467.5 Caspase Martin U. (2007) Apoptosis 12 525 Misaghi S. (2004) Chem. Biol. 11 1677 WO2001058526 Merck (Calbiochem) Download

Results as Barchart

View results as a bar chart
3µM

Results as Table

Screening Concentration: 3µM
Kinase % Activity Remainingsort descending Standard Deviation
Src 10 1
Lck 10 1
S6K1 33 2
MNK1 42 2
CAMKK beta 49 3
BRSK2 53 6
CSK 55 7
PIM3 56 6
ERK8 58 4
Aurora B 59 3
PIM1 61 6
CK1 delta 63 6
MNK2 65 6
MELK 65 8
GSK3 beta 65 6
DYRK3 68 7
CAMKK alpha 70 12
p38 alpha MAPK 72 2
RSK2 74 2
Aurora C 75 6
MSK1 75 3
MST2 76 4
CAMK1 77 9
AMPK 79 4
HIPK2 79 11
HIPK3 79 9
ERK2 79 5
MARK3 80 3
MKK1 80 8
CDK2-Cyclin A 80 7
JNK1 81 3
CHK2 81 9
PKB alpha 82 3
SmMLCK 82 4
PLK1 82 5
JNK2 83 5
PRK2 83 3
PKD1 83 4
SRPK1 85 1
PKA 85 7
PKC alpha 85 7
p38 beta MAPK 85 4
PIM2 85 10
DYRK1A 86 11
ROCK 2 86 7
PAK5 88 6
CHK1 88 4
PDK1 89 10
JNK3 89 4
NEK6 90 4
PAK4 91 1
DYRK2 91 8
PKC zeta 91 5
RSK1 92 6
MAPKAP-K3 92 6
CK2 92 10
ERK1 92 6
NEK7 92 8
IKK beta 92 8
p38 gamma MAPK 92 7
PAK6 93 5
PHK 93 5
MAPKAP-K2 94 10
NEK2a 95 4
EF2K 97 8
PRAK 97 5
PKB beta 97 4
p38 delta MAPK 103 9
SGK1 107 8

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