Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
FMK (Caspase Inhibitor I) C22H30FN3O7 467.5 Caspase Martin U. (2007) Apoptosis 12 525 Misaghi S. (2004) Chem. Biol. 11 1677 WO2001058526 Merck (Calbiochem) Download

Results as Barchart

View results as a bar chart
3µM

Results as Table

Screening Concentration: 3µM
Kinase % Activity Remaining Standard Deviation
MKK1 80 8
ERK1 92 6
ERK2 79 5
JNK1 81 3
JNK2 83 5
JNK3 89 4
p38 alpha MAPK 72 2
p38 beta MAPK 85 4
p38 gamma MAPK 92 7
p38 delta MAPK 103 9
ERK8 58 4
RSK1 92 6
RSK2 74 2
PDK1 89 10
PKB alpha 82 3
PKB beta 97 4
SGK1 107 8
S6K1 33 2
PKA 85 7
ROCK 2 86 7
PRK2 83 3
PKC alpha 85 7
PKC zeta 91 5
PKD1 83 4
MSK1 75 3
MNK1 42 2
MNK2 65 6
MAPKAP-K2 94 10
MAPKAP-K3 92 6
PRAK 97 5
CAMKK alpha 70 12
CAMKK beta 49 3
CAMK1 77 9
SmMLCK 82 4
PHK 93 5
CHK1 88 4
CHK2 81 9
GSK3 beta 65 6
CDK2-Cyclin A 80 7
PLK1 82 5
Aurora B 59 3
Aurora C 75 6
AMPK 79 4
MARK3 80 3
BRSK2 53 6
MELK 65 8
CK1 delta 63 6
CK2 92 10
DYRK1A 86 11
DYRK2 91 8
DYRK3 68 7
NEK2a 95 4
NEK6 90 4
NEK7 92 8
IKK beta 92 8
PIM1 61 6
PIM2 85 10
PIM3 56 6
SRPK1 85 1
EF2K 97 8
HIPK2 79 11
HIPK3 79 9
PAK4 91 1
PAK5 88 6
PAK6 93 5
MST2 76 4
Src 10 1
Lck 10 1
CSK 55 7

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