Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
EGCG (Epigallocatechin Gallate) C22H18O11 458.4 PKC Dell'Aica I. (2004) EMBO Rep. 5 418-422 Tachibana H. (2004) Nat. Struct. Mol. Biol. 11 380 WO2001051048 Merck (Calbiochem) Download

Results as Barchart

View results as a bar chart
10µM

Results as Table

Screening Concentration: 10µM
Kinase % Activity Remainingsort descending Standard Deviation
DYRK2 0 1
EPH-B3 1 0
PKB beta 1 0
PKC zeta 2 1
SRPK1 5 3
PRAK 5 2
DYRK3 5 0
NEK2a 5 1
MARK3 6 1
RSK2 6 6
DYRK1A 6 0
FGF-R1 6 0
PLK1 7 2
PAK6 8 4
YES1 12 3
Aurora B 12 3
PIM1 15 2
HIPK2 15 0
PKD1 16 1
ERK1 17 1
PIM3 17 0
BTK 18 0
IGF-1R 19 4
CAMK1 19 8
VEGFR1 20 1
ERK8 20 0
IKK beta 21 3
Src 21 0
PAK4 22 1
MAPKAP-K2 22 1
BRSK2 23 1
MST4 24 1
IKK epsilon 27 4
IRR 28 1
PAK5 35 1
S6K1 37 1
MST2 37 0
MSK1 40 4
RSK1 46 2
PIM2 47 0
SmMLCK 51 2
MELK 53 1
NEK6 56 4
MKK1 58 24
SGK1 58 2
CHK2 61 1
TBK1 65 4
CAMKK beta 65 2
AMPK 66 2
SYK 67 8
GSK3 beta 70 6
IR 70 5
MNK1 71 10
CHK1 72 3
ERK2 72 4
MNK2 73 7
PDK1 73 0
ROCK 2 74 5
PKB alpha 75 20
PHK 75 6
EPH-A2 76 0
p38 alpha MAPK 80 8
PKC alpha 81 3
PRK2 82 3
JNK2 84 2
EF2K 86 2
PKA 87 1
CDK2-Cyclin A 88 4
CSK 88 10
CK2 89 17
CK1 delta 90 9
Lck 90 3
p38 beta MAPK 96 20
p38 gamma MAPK 98 15
p38 delta MAPK 102 17
JNK1 106 8

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