InhibitorScreening ConcentrationKinase% Activity RemainingStandard Deviation
BX-517 Analog (compound 7b)0.10µMMKK181
BX-517 Analog (compound 7b)0.10µMERK1717
BX-517 Analog (compound 7b)0.10µMERK28110
BX-517 Analog (compound 7b)0.10µMJNK11241
BX-517 Analog (compound 7b)0.10µMJNK2214172
BX-517 Analog (compound 7b)0.10µMp38 alpha MAPK818
BX-517 Analog (compound 7b)0.10µMp38 beta MAPK1030
BX-517 Analog (compound 7b)0.10µMp38 gamma MAPK936
BX-517 Analog (compound 7b)0.10µMp38 delta MAPK859
BX-517 Analog (compound 7b)0.10µMERK850
BX-517 Analog (compound 7b)0.10µMRSK1244
BX-517 Analog (compound 7b)0.10µMRSK2384
BX-517 Analog (compound 7b)0.10µMPDK1201
BX-517 Analog (compound 7b)0.10µMPKB alpha 854
BX-517 Analog (compound 7b)0.10µMPKB beta 883
BX-517 Analog (compound 7b)0.10µMSGK1775
BX-517 Analog (compound 7b)0.10µMS6K1760
BX-517 Analog (compound 7b)0.10µMPKA780
BX-517 Analog (compound 7b)0.10µMROCK 210325
BX-517 Analog (compound 7b)0.10µMPRK22511
BX-517 Analog (compound 7b)0.10µMPKC alpha 1063
BX-517 Analog (compound 7b)0.10µMPKC zeta 854
BX-517 Analog (compound 7b)0.10µMPKD1302
BX-517 Analog (compound 7b)0.10µMMSK1981
BX-517 Analog (compound 7b)0.10µMMNK1800
BX-517 Analog (compound 7b)0.10µMMNK27512
BX-517 Analog (compound 7b)0.10µMMAPKAP-K2 863
BX-517 Analog (compound 7b)0.10µMPRAK956
BX-517 Analog (compound 7b)0.10µMCAMKK beta 677
BX-517 Analog (compound 7b)0.10µMCAMK111212
BX-517 Analog (compound 7b)0.10µMSmMLCK547
BX-517 Analog (compound 7b)0.10µMPHK130
BX-517 Analog (compound 7b)0.10µMCHK1852
BX-517 Analog (compound 7b)0.10µMCHK2-10
BX-517 Analog (compound 7b)0.10µMGSK3 beta 111
BX-517 Analog (compound 7b)0.10µMCDK2-Cyclin A630
BX-517 Analog (compound 7b)0.10µMPLK1865
BX-517 Analog (compound 7b)0.10µMAMPK50
BX-517 Analog (compound 7b)0.10µMMARK3163
BX-517 Analog (compound 7b)0.10µMBRSK2133
BX-517 Analog (compound 7b)0.10µMMELK160
BX-517 Analog (compound 7b)0.10µMCK1 delta 900
BX-517 Analog (compound 7b)0.10µMCK29317
BX-517 Analog (compound 7b)0.10µMDYRK1A429
BX-517 Analog (compound 7b)0.10µMDYRK2193
BX-517 Analog (compound 7b)0.10µMDYRK3193
BX-517 Analog (compound 7b)0.10µMNEK2a10010
BX-517 Analog (compound 7b)0.10µMNEK6926
BX-517 Analog (compound 7b)0.10µMIKK beta 751
BX-517 Analog (compound 7b)0.10µMIKK epsilon 5114
BX-517 Analog (compound 7b)0.10µMTBK12717
BX-517 Analog (compound 7b)0.10µMPIM1432
BX-517 Analog (compound 7b)0.10µMPIM2766
BX-517 Analog (compound 7b)0.10µMPIM3300
BX-517 Analog (compound 7b)0.10µMSRPK1904
BX-517 Analog (compound 7b)0.10µMEF2K10214
BX-517 Analog (compound 7b)0.10µMHIPK2331
BX-517 Analog (compound 7b)0.10µMPAK4645
BX-517 Analog (compound 7b)0.10µMPAK57510
BX-517 Analog (compound 7b)0.10µMPAK6861
BX-517 Analog (compound 7b)0.10µMMST280
BX-517 Analog (compound 7b)0.10µMMST45532
BX-517 Analog (compound 7b)0.10µMSrc412
BX-517 Analog (compound 7b)0.10µMLck444
BX-517 Analog (compound 7b)0.10µMCSK980
BX-517 Analog (compound 7b)0.10µMYES1324
BX-517 Analog (compound 7b)0.10µMBTK8611
BX-517 Analog (compound 7b)0.10µMSYK9523
BX-517 Analog (compound 7b)0.10µMEPH-A2930
BX-517 Analog (compound 7b)0.10µMEPH-B31071
BX-517 Analog (compound 7b)0.10µMFGF-R1173
BX-517 Analog (compound 7b)0.10µMIGF-1R4949
BX-517 Analog (compound 7b)0.10µMIR11214
BX-517 Analog (compound 7b)0.10µMIRR350
BX-517 Analog (compound 7b)0.10µMVEGFR170
BX-517 Analog (compound 7b)1.00µMMKK110
BX-517 Analog (compound 7b)1.00µMERK16052
BX-517 Analog (compound 7b)1.00µMERK2419
BX-517 Analog (compound 7b)1.00µMJNK1991
BX-517 Analog (compound 7b)1.00µMJNK2430
BX-517 Analog (compound 7b)1.00µMp38 alpha MAPK804
BX-517 Analog (compound 7b)1.00µMp38 beta MAPK805
BX-517 Analog (compound 7b)1.00µMp38 gamma MAPK864
BX-517 Analog (compound 7b)1.00µMp38 delta MAPK621
BX-517 Analog (compound 7b)1.00µMERK820
BX-517 Analog (compound 7b)1.00µMRSK1104
BX-517 Analog (compound 7b)1.00µMRSK23214
BX-517 Analog (compound 7b)1.00µMPDK130
BX-517 Analog (compound 7b)1.00µMPKB alpha 690
BX-517 Analog (compound 7b)1.00µMPKB beta 777
BX-517 Analog (compound 7b)1.00µMSGK1320
BX-517 Analog (compound 7b)1.00µMS6K1320
BX-517 Analog (compound 7b)1.00µMPKA660
BX-517 Analog (compound 7b)1.00µMROCK 2374
BX-517 Analog (compound 7b)1.00µMPRK253
BX-517 Analog (compound 7b)1.00µMPKC alpha 835
BX-517 Analog (compound 7b)1.00µMPKC zeta 661
BX-517 Analog (compound 7b)1.00µMPKD130
BX-517 Analog (compound 7b)1.00µMMSK1732
BX-517 Analog (compound 7b)1.00µMMNK1540
BX-517 Analog (compound 7b)1.00µMMNK2465
BX-517 Analog (compound 7b)1.00µMMAPKAP-K2 496
BX-517 Analog (compound 7b)1.00µMPRAK506
BX-517 Analog (compound 7b)1.00µMCAMKK beta 4112
BX-517 Analog (compound 7b)1.00µMCAMK1695
BX-517 Analog (compound 7b)1.00µMSmMLCK111
BX-517 Analog (compound 7b)1.00µMPHK10
BX-517 Analog (compound 7b)1.00µMCHK140
BX-517 Analog (compound 7b)1.00µMCHK2-50
BX-517 Analog (compound 7b)1.00µMGSK3 beta 73
BX-517 Analog (compound 7b)1.00µMCDK2-Cyclin A142
BX-517 Analog (compound 7b)1.00µMPLK1424
BX-517 Analog (compound 7b)1.00µMAMPK64
BX-517 Analog (compound 7b)1.00µMMARK351
BX-517 Analog (compound 7b)1.00µMBRSK2103
BX-517 Analog (compound 7b)1.00µMMELK30
BX-517 Analog (compound 7b)1.00µMCK1 delta 5910
BX-517 Analog (compound 7b)1.00µMCK2655
BX-517 Analog (compound 7b)1.00µMDYRK1A116
BX-517 Analog (compound 7b)1.00µMDYRK220
BX-517 Analog (compound 7b)1.00µMDYRK341
BX-517 Analog (compound 7b)1.00µMNEK2a752
BX-517 Analog (compound 7b)1.00µMNEK67610
BX-517 Analog (compound 7b)1.00µMIKK beta 7527
BX-517 Analog (compound 7b)1.00µMIKK epsilon 121
BX-517 Analog (compound 7b)1.00µMTBK176
BX-517 Analog (compound 7b)1.00µMPIM190
BX-517 Analog (compound 7b)1.00µMPIM2340
BX-517 Analog (compound 7b)1.00µMPIM392
BX-517 Analog (compound 7b)1.00µMSRPK1751
BX-517 Analog (compound 7b)1.00µMEF2K863
BX-517 Analog (compound 7b)1.00µMHIPK270
BX-517 Analog (compound 7b)1.00µMPAK4310
BX-517 Analog (compound 7b)1.00µMPAK5430
BX-517 Analog (compound 7b)1.00µMPAK6773
BX-517 Analog (compound 7b)1.00µMMST221
BX-517 Analog (compound 7b)1.00µMMST4180
BX-517 Analog (compound 7b)1.00µMSrc70
BX-517 Analog (compound 7b)1.00µMLck100
BX-517 Analog (compound 7b)1.00µMCSK696
BX-517 Analog (compound 7b)1.00µMYES180
BX-517 Analog (compound 7b)1.00µMBTK295
BX-517 Analog (compound 7b)1.00µMSYK401
BX-517 Analog (compound 7b)1.00µMEPH-A2545
BX-517 Analog (compound 7b)1.00µMEPH-B39011
BX-517 Analog (compound 7b)1.00µMFGF-R120
BX-517 Analog (compound 7b)1.00µMIGF-1R337
BX-517 Analog (compound 7b)1.00µMIR10111
BX-517 Analog (compound 7b)1.00µMIRR165
BX-517 Analog (compound 7b)1.00µMVEGFR131
BX-517 Analog (compound 7b)10.00µMMKK121
BX-517 Analog (compound 7b)10.00µMERK140
BX-517 Analog (compound 7b)10.00µMERK2163
BX-517 Analog (compound 7b)10.00µMJNK1484
BX-517 Analog (compound 7b)10.00µMJNK2170
BX-517 Analog (compound 7b)10.00µMp38 alpha MAPK456
BX-517 Analog (compound 7b)10.00µMp38 beta MAPK499
BX-517 Analog (compound 7b)10.00µMp38 gamma MAPK7527
BX-517 Analog (compound 7b)10.00µMp38 delta MAPK221
BX-517 Analog (compound 7b)10.00µMERK810
BX-517 Analog (compound 7b)10.00µMRSK150
BX-517 Analog (compound 7b)10.00µMRSK2223
BX-517 Analog (compound 7b)10.00µMPDK102
BX-517 Analog (compound 7b)10.00µMPKB alpha 627
BX-517 Analog (compound 7b)10.00µMPKB beta 364
BX-517 Analog (compound 7b)10.00µMSGK162
BX-517 Analog (compound 7b)10.00µMS6K1121
BX-517 Analog (compound 7b)10.00µMPKA325
BX-517 Analog (compound 7b)10.00µMROCK 271
BX-517 Analog (compound 7b)10.00µMPRK260
BX-517 Analog (compound 7b)10.00µMPKC alpha 277
BX-517 Analog (compound 7b)10.00µMPKC zeta 214
BX-517 Analog (compound 7b)10.00µMPKD132
BX-517 Analog (compound 7b)10.00µMMSK1300
BX-517 Analog (compound 7b)10.00µMMNK13014
BX-517 Analog (compound 7b)10.00µMMNK2162
BX-517 Analog (compound 7b)10.00µMMAPKAP-K2 106
BX-517 Analog (compound 7b)10.00µMPRAK81
BX-517 Analog (compound 7b)10.00µMCAMKK beta 353
BX-517 Analog (compound 7b)10.00µMCAMK1190
BX-517 Analog (compound 7b)10.00µMSmMLCK11
BX-517 Analog (compound 7b)10.00µMPHK00
BX-517 Analog (compound 7b)10.00µMCHK110
BX-517 Analog (compound 7b)10.00µMCHK214
BX-517 Analog (compound 7b)10.00µMGSK3 beta 32
BX-517 Analog (compound 7b)10.00µMCDK2-Cyclin A60
BX-517 Analog (compound 7b)10.00µMPLK1186
BX-517 Analog (compound 7b)10.00µMAMPK41
BX-517 Analog (compound 7b)10.00µMMARK331
BX-517 Analog (compound 7b)10.00µMBRSK2183
BX-517 Analog (compound 7b)10.00µMMELK00
BX-517 Analog (compound 7b)10.00µMCK1 delta 205
BX-517 Analog (compound 7b)10.00µMCK2211
BX-517 Analog (compound 7b)10.00µMDYRK1A2733
BX-517 Analog (compound 7b)10.00µMDYRK200
BX-517 Analog (compound 7b)10.00µMDYRK310
BX-517 Analog (compound 7b)10.00µMNEK2a281
BX-517 Analog (compound 7b)10.00µMNEK6382
BX-517 Analog (compound 7b)10.00µMIKK beta 264
BX-517 Analog (compound 7b)10.00µMIKK epsilon 116
BX-517 Analog (compound 7b)10.00µMTBK1119
BX-517 Analog (compound 7b)10.00µMPIM122
BX-517 Analog (compound 7b)10.00µMPIM280
BX-517 Analog (compound 7b)10.00µMPIM372
BX-517 Analog (compound 7b)10.00µMSRPK1363
BX-517 Analog (compound 7b)10.00µMEF2K1167
BX-517 Analog (compound 7b)10.00µMHIPK210
BX-517 Analog (compound 7b)10.00µMPAK42931
BX-517 Analog (compound 7b)10.00µMPAK580
BX-517 Analog (compound 7b)10.00µMPAK6384
BX-517 Analog (compound 7b)10.00µMMST200
BX-517 Analog (compound 7b)10.00µMMST4216
BX-517 Analog (compound 7b)10.00µMSrc10
BX-517 Analog (compound 7b)10.00µMLck30
BX-517 Analog (compound 7b)10.00µMCSK426
BX-517 Analog (compound 7b)10.00µMYES131
BX-517 Analog (compound 7b)10.00µMBTK96
BX-517 Analog (compound 7b)10.00µMSYK70
BX-517 Analog (compound 7b)10.00µMEPH-A2201
BX-517 Analog (compound 7b)10.00µMEPH-B3538
BX-517 Analog (compound 7b)10.00µMFGF-R110
BX-517 Analog (compound 7b)10.00µMIGF-1R10
BX-517 Analog (compound 7b)10.00µMIR266
BX-517 Analog (compound 7b)10.00µMIRR52
BX-517 Analog (compound 7b)10.00µMVEGFR110