Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
Blebbistatin C18H16N2O2 292.3 myosin II Shu S. (2005) Proc. Natl. Acad. Sci. USA 102 1472 Kovacs M. (2004) J. Biol. Chem. 279 35557 WO2012062819 Merck (Calbiochem) Download

Results as Barchart

View results as a bar chart
100µM
10µM

Results as Table

Screening Concentration: 100µM
Kinase % Activity Remainingsort descending Standard Deviation
SGK1 60 3
AMPK 60 2
PRAK 64 1
GSK3 beta 66 2
CSK 67 9
PKA 70 0
S6K1 71 4
p38 beta MAPK 71 7
Lck 72 1
PDK1 74 3
PKC alpha 75 7
MSK1 75 7
ROCK 2 76 0
RSK1 77 5
JNK1 78 5
MAPKAP-K2 80 4
p38 alpha MAPK 80 1
p38 gamma MAPK 80 0
NEK2a 82 6
ERK2 82 3
NEK6 85 2
PHK 86 2
PKB alpha 88 3
DYRK1A 90 3
CK1 delta 91 3
CDK2-Cyclin A 92 7
CHK1 96 7
MKK1 99 6
CK2 101 5
p38 delta MAPK 116 4
Screening Concentration: 10µM
Kinase % Activity Remainingsort descending Standard Deviation
CSK 69 7
RSK2 72 3
MINK1 72 9
PAK5 73 7
MLK3 73 7
PKB beta 74 6
CAMK1 74 4
SmMLCK 74 15
RSK1 76 1
DYRK2 76 10
NEK2a 77 2
ROCK 2 77 4
Src 80 6
p38 delta MAPK 81 1
LKB1 81 1
MKK2 81 13
MAPKAP-K2 82 4
BTK 82 9
PRAK 82 3
TAO1 82 5
p38 beta MAPK 82 1
PAK6 83 6
PIM3 83 7
EF2K 83 5
MSK1 83 0
VEGFR1 85 2
IKK epsilon 85 6
MAPKAP-K3 86 1
IRAK4 86 6
PIM1 87 6
CLK2 87 5
HER4 87 8
PAK2 87 5
TTK 87 3
Aurora B 88 2
IRR 88 7
SRPK1 88 1
HIPK1 88 5
JNK2 88 6
GSK3 beta 88 0
IGF-1R 88 2
ERK8 89 5
MKK1 89 6
CAMKK beta 90 3
CHK1 90 5
RIPK2 90 7
PAK4 90 8
MARK3 91 4
ERK2 91 9
ASK1 91 3
AMPK 92 8
S6K1 92 3
JNK1 92 2
PDK1 93 3
MARK2 93 1
PIM2 93 3
DAPK1 93 1
TBK1 94 6
MARK4 94 5
MKK6 94 0
PKB alpha 95 1
PRK2 95 0
IR 95 15
IKK beta 96 4
YES1 96 2
MARK1 96 2
MELK 96 3
TAK1 96 3
MNK1 97 2
GCK 97 8
EPH-B1 97 11
NUAK1 97 3
DYRK1A 97 4
PKD1 97 11
BRSK2 98 4
HIPK2 98 0
MST4 99 1
CK1 delta 99 4
EPH-B4 99 2
JNK3 99 2
PLK1 99 8
p38 gamma MAPK 99 2
Aurora A 99 3
DYRK3 99 9
MEKK1 100 8
CHK2 100 12
JAK2 101 13
SGK1 101 0
MLK1 101 8
PKA 101 6
p38 alpha MAPK 101 2
ERK1 102 1
TrkA 103 3
PKC alpha 103 4
HIPK3 103 5
MNK2 104 3
MST2 104 1
SYK 105 12
Lck 106 6
BRSK1 106 5
NEK6 107 4
EPH-B3 107 4
EPH-A4 108 13
PKC zeta 108 5
EPH-A2 109 8
CK2 110 5
PHK 114 0
EPH-B2 116 3
CDK2-Cyclin A 116 1
FGF-R1 118 14

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