Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
ARA014418 C12H12N4O4S 308.3 GSK3 Noble W. (2005) Proc. Natl. Acad. Sci. USA 102 6990 Bhat R. (2003) J. Biol. Chem. 278 45937 WO2013124413 Sigma Download

Results as Barchart

View results as a bar chart
10µM

Results as Table

Screening Concentration: 10µM
Kinase % Activity Remainingsort ascending Standard Deviation
YES1 111 7
p38 alpha MAPK 109 8
SYK 107 10
MAPKAP-K2 103 2
p38 beta MAPK 102 8
ERK1 101 1
EPH-A2 101 5
MST4 99 14
EF2K 98 5
NEK7 96 2
PKB alpha 95 2
ERK2 94 7
MNK2 94 5
CHK2 93 2
PKD1 92 4
PIM2 92 5
NEK6 91 1
JNK3 91 0
FGF-R1 91 8
SmMLCK 90 2
PHK 90 4
p38 gamma MAPK 89 1
CK1 delta 89 6
HIPK3 88 1
SGK1 87 3
PRK2 85 2
PKB beta 85 2
Aurora C 84 3
RSK2 84 1
ROCK 2 83 2
CHK1 83 2
PIM1 83 3
IKK epsilon 83 3
CSK 82 2
DYRK2 81 7
Src 81 1
NEK2a 81 2
MAPKAP-K3 81 4
JNK1 80 1
Lck 80 1
PKC alpha 80 3
MSK1 80 4
p38 delta MAPK 80 2
MNK1 80 2
MST2 80 7
RSK1 79 4
CAMKK alpha 79 5
CK2 79 1
PLK1 78 0
TBK1 78 2
MKK1 77 9
CAMK1 76 3
PAK5 76 0
BRSK2 76 4
S6K1 75 2
IKK beta 75 3
MARK3 75 4
MELK 75 4
PAK6 74 2
SRPK1 74 5
PDK1 74 1
CAMKK beta 73 9
JNK2 72 5
AMPK 72 1
DYRK3 71 1
Aurora B 71 3
PKC zeta 70 1
PIM3 69 0
PKA 68 4
PRAK 67 5
PAK4 66 2
HIPK2 53 3
DYRK1A 50 6
IRR 45 1
ERK8 37 3
CDK2-Cyclin A 23 2
GSK3 beta 3 0

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