Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
ARA014418 C12H12N4O4S 308.3 GSK3 Noble W. (2005) Proc. Natl. Acad. Sci. USA 102 6990 Bhat R. (2003) J. Biol. Chem. 278 45937 WO2013124413 Sigma Download

Results as Barchart

View results as a bar chart
10µM

Results as Table

Screening Concentration: 10µM
Kinase % Activity Remainingsort descending Standard Deviation
GSK3 beta 3 0
CDK2-Cyclin A 23 2
ERK8 37 3
IRR 45 1
DYRK1A 50 6
HIPK2 53 3
PAK4 66 2
PRAK 67 5
PKA 68 4
PIM3 69 0
PKC zeta 70 1
DYRK3 71 1
Aurora B 71 3
AMPK 72 1
JNK2 72 5
CAMKK beta 73 9
SRPK1 74 5
PDK1 74 1
PAK6 74 2
MARK3 75 4
MELK 75 4
S6K1 75 2
IKK beta 75 3
BRSK2 76 4
CAMK1 76 3
PAK5 76 0
MKK1 77 9
TBK1 78 2
PLK1 78 0
RSK1 79 4
CAMKK alpha 79 5
CK2 79 1
p38 delta MAPK 80 2
MNK1 80 2
MST2 80 7
JNK1 80 1
Lck 80 1
PKC alpha 80 3
MSK1 80 4
MAPKAP-K3 81 4
DYRK2 81 7
Src 81 1
NEK2a 81 2
CSK 82 2
IKK epsilon 83 3
ROCK 2 83 2
CHK1 83 2
PIM1 83 3
Aurora C 84 3
RSK2 84 1
PKB beta 85 2
PRK2 85 2
SGK1 87 3
HIPK3 88 1
CK1 delta 89 6
p38 gamma MAPK 89 1
SmMLCK 90 2
PHK 90 4
NEK6 91 1
JNK3 91 0
FGF-R1 91 8
PKD1 92 4
PIM2 92 5
CHK2 93 2
MNK2 94 5
ERK2 94 7
PKB alpha 95 2
NEK7 96 2
EF2K 98 5
MST4 99 14
ERK1 101 1
EPH-A2 101 5
p38 beta MAPK 102 8
MAPKAP-K2 103 2
SYK 107 10
p38 alpha MAPK 109 8
YES1 111 7

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