Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
ARA014418 C12H12N4O4S 308.3 GSK3 Noble W. (2005) Proc. Natl. Acad. Sci. USA 102 6990 Bhat R. (2003) J. Biol. Chem. 278 45937 WO2013124413 Sigma Download

Results as Barchart

View results as a bar chart
10µM

Results as Table

Screening Concentration: 10µM
Kinase % Activity Remaining Standard Deviation
MKK1 77 9
ERK1 101 1
ERK2 94 7
JNK1 80 1
JNK2 72 5
JNK3 91 0
p38 alpha MAPK 109 8
p38 beta MAPK 102 8
p38 gamma MAPK 89 1
p38 delta MAPK 80 2
ERK8 37 3
RSK1 79 4
RSK2 84 1
PDK1 74 1
PKB alpha 95 2
PKB beta 85 2
SGK1 87 3
S6K1 75 2
PKA 68 4
ROCK 2 83 2
PRK2 85 2
PKC alpha 80 3
PKC zeta 70 1
PKD1 92 4
MSK1 80 4
MNK1 80 2
MNK2 94 5
MAPKAP-K2 103 2
MAPKAP-K3 81 4
PRAK 67 5
CAMKK alpha 79 5
CAMKK beta 73 9
CAMK1 76 3
SmMLCK 90 2
PHK 90 4
CHK1 83 2
CHK2 93 2
GSK3 beta 3 0
CDK2-Cyclin A 23 2
PLK1 78 0
Aurora B 71 3
Aurora C 84 3
AMPK 72 1
MARK3 75 4
BRSK2 76 4
MELK 75 4
CK1 delta 89 6
CK2 79 1
DYRK1A 50 6
DYRK2 81 7
DYRK3 71 1
NEK2a 81 2
NEK6 91 1
NEK7 96 2
IKK beta 75 3
IKK epsilon 83 3
TBK1 78 2
PIM1 83 3
PIM2 92 5
PIM3 69 0
SRPK1 74 5
EF2K 98 5
HIPK2 53 3
HIPK3 88 1
PAK4 66 2
PAK5 76 0
PAK6 74 2
MST2 80 7
MST4 99 14
Src 81 1
Lck 80 1
CSK 82 2
YES1 111 7
SYK 107 10
EPH-A2 101 5
FGF-R1 91 8
IRR 45 1

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