Kinase Profiling Inhibitor Database

Inhibitor Structure Image Brutto MW Action Reference Reference 2 Patent Commercial Vendor Notes Results
CCT250862 NEK Download

Results as Barchart

View results as a bar chart
1µM

Results as Table

Screening Concentration: 1µM
Kinase % Activity Remainingsort ascending Standard Deviation
EPH-B1 114 10
Aurora A 113 5
p38 alpha MAPK 108 24
WNK1 108 8
NEK6 106 3
CAMK1 105 2
MPSK1 100 1
EIF2AK3 100 2
MAPKAP-K3 99 0
TTBK1 98 12
PAK5 97 10
TLK1 96 3
CK2 96 8
PAK6 95 3
ZAP70 95 14
PIM2 95 2
PKB beta 95 25
SYK 94 1
EPH-B4 94 11
TTBK2 94 3
HER4 93 4
DYRK2 92 6
IKK beta 91 4
MAPKAP-K2 91 3
MKK2 91 3
EPH-B3 91 14
p38 gamma MAPK 90 6
PKB alpha 89 2
PRAK 89 5
ROCK 2 89 10
PAK2 87 6
p38 beta MAPK 86 5
PKA 86 4
JNK3 86 10
EF2K 85 4
MEKK1 85 2
CHK1 85 3
MKK1 84 3
PAK4 84 1
MKK6 82 7
PLK1 81 17
DAPK1 81 6
p38 delta MAPK 80 0
SRPK1 78 3
ERK1 78 3
TESK1 76 11
JNK1 76 2
PDK1 74 10
ERK2 74 6
ASK1 73 11
PDGFRA 70 11
JNK2 70 3
EPH-A2 69 2
PKC zeta 68 9
OSR1 68 5
BRK 68 4
ULK1 67 8
HIPK3 65 14
EPH-A4 64 13
IR 64 8
TTK 62 1
RSK2 62 1
MST3 60 2
SIK3 56 0
CSK 55 2
NEK2a 55 15
CDK9-Cyclin T1 54 9
Aurora B 54 16
SGK1 54 2
CHK2 51 5
TSSK1 51 1
PIM3 51 3
PIM1 48 5
LKB1 46 3
MARK1 46 3
MARK4 45 7
TBK1 42 10
RSK1 42 16
TGFBR1 42 1
CDK2-Cyclin A 41 7
TIE2 41 1
MST4 41 11
EPH-B2 40 5
CK1 gamma 2 39 5
CAMKK beta 38 44
DYRK3 38 2
MNK1 37 8
ULK2 37 3
BTK 37 3
PKC gamma 36 6
ERK5 36 7
MARK2 34 3
IRAK4 33 7
IKK epsilon 32 3
PKC alpha 32 3
PKD1 31 2
HIPK1 30 12
MSK1 29 5
DDR2 28 2
MELK 27 5
JAK2 27 0
MARK3 26 1
STK33 25 2
MNK2 25 2
TAO1 25 0
AMPK 24 4
PHK 24 0
MST2 23 11
HIPK2 23 6
BRSK1 23 6
BRSK2 21 2
S6K1 21 2
SmMLCK 18 2
MLK1 17 7
FGF-R1 17 1
IGF-1R 17 7
ABL 17 1
PRK2 17 1
IRR 16 2
ERK8 15 7
AMPK (hum) 15 2
SIK2 14 5
Src 13 1
RIPK2 11 2
IRAK1 11 3
TrkA 10 1
CK1 delta 9 1
Lck 9 1
MAP4K5 7 1
VEGFR1 6 0
MAP4K3 6 2
MINK1 6 1
YES1 6 1
TAK1 6 0
GSK3 beta 5 1
MLK3 4 1
DYRK1A 4 0
GCK 3 0
NUAK1 2 1
CLK2 2 0

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